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GPCR

Use of Backbone Modification To Enlarge the Spatiotemporal Diversity of Parathyroid Hormone Receptor‑1 Signaling via Biased Agonism

Posted on June 27, 2022

Use of Backbone Modification To Enlarge the Spatiotemporal diversity of Parathyroid Hormone Receptor‑1 Signaling via Biased Agonism

File: Use-of-Backbone-Modification-jacs.9b04179.pdf

Impact of substitution registry on receptor-activation profiles of backbone-modified glucagon-like peptide-1 analogues

Posted on June 27, 2022

Impact of substitution registry on receptor-activation profiles of backbone-modified glucagon-like peptide-1 analogues

File: Impact-of-substitution-nihms-1053525.pdf

Spatial bias in cAMP generation determines biological responses to PTH type 1 receptor activation

Posted on June 27, 2022

Spatial bias in cAMP generation determines biological responses to PTH type 1 receptor activation

File: Spatial-bias-nihms-1761601.pdf

Structural and functional diversity among agonist-bound states of the GLP-1 receptor

Posted on June 27, 2022

Structural and functional diversity among agonist-bound states of the GLP-1 receptor

File: Structural-and-functional-diversity-s41589-021-00945-w.pdf

β‐Arrestin-Biased Agonists of the GLP‐1 Receptor from β‐Amino Acid Residue Incorporation into GLP‐1 Analogues

Posted on August 10, 2020

β‐Arrestin-Biased Agonists of the GLP‐1 Receptor from β‐Amino Acid Residue Incorporation into GLP‐1 Analogues

File: Hager-biased-ag-JACS-16.pdf

Backbone modification of a polypeptide drug alters duration of action in vivo

Posted on August 10, 2020

Backbone modification of a polypeptide drug alters duration of action in vivo

File: Cheloha-PTH-NBT-14.pdf

Receptor selectivity from minimal backbone modification of a polypeptide agonist

Posted on August 10, 2020

Receptor selectivity from minimal backbone modification of a polypeptide agonist

File: Liu-Shi-R1-vs.-R2-18.pdf

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